Basic Information
ID: ALA4815613
Type: Binding
Description: Displacement of [3H]-NMS from human muscarinic M5 receptor expressed in CHO cell membranes assessed as inhibition constant by radioligand competition analysis
Organism: Homo sapiens
Cell type: CHO
Subcellular Fraction: Cell membrane
Activity Charts
Bioactivity
Activity Types for Assay ALA4815613
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 627.79 | 4.27 | 4.27 |
| 552.14 | 5.31 | 5.31 |
| 732.93 | 2.30 | 2.30 |
| 869.04 | 5.08 | 5.08 |
| 916.19 | 1.42 | 1.42 |
| 961.88 | -1.00 | -1.00 |
| 1230.98 | 1.73 | 1.73 |
| 1386.26 | 0.95 | 0.95 |
| 1473.21 | -1.27 | -1.27 |
| 1501.27 | -0.51 | -0.51 |
| 1358.20 | 0.17 | 0.17 |
| 1458.24 | 0.64 | 0.64 |
| 1060.97 | 1.91 | 1.91 |
| 1444.21 | 0.25 | 0.25 |
| 1459.19 | -1.66 | -1.66 |
| 1501.27 | -0.49 | -0.49 |
| 1358.20 | 0.17 | 0.17 |
| 1472.27 | 1.03 | 1.03 |
| 1416.16 | -0.39 | -0.39 |
| 1117.98 | -0.48 | -0.48 |
| 1487.24 | -0.88 | -0.88 |
| 1473.21 | -1.27 | -1.27 |
| 1372.23 | 0.56 | 0.56 |
| 1487.24 | -0.88 | -0.88 |
| 1458.24 | 0.64 | 0.64 |
| 1473.21 | -1.27 | -1.27 |
| 1258.21 | 0.56 | 0.56 |
| 1401.19 | 1.52 | 1.52 |
| 1344.18 | -0.22 | -0.22 |