Basic Information
ID: ALA4815931
Type: Binding
Description: Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Dual specificty protein kinase CLK1(ALA4224)
Document: ALA4813966
Inhibition of recombinant human CLK1 (130 to end residues) using ERMRPRKRQGSVR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4815931
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 361.41 | 2.67 | 2.67 |
| 436.52 | 5.27 | 5.27 |
| 407.47 | 5.09 | 5.09 |
| 345.41 | 3.23 | 3.23 |
| 331.38 | 2.66 | 2.66 |
| 422.49 | 4.88 | 4.88 |
| 408.46 | 4.49 | 4.49 |
| 361.41 | 2.67 | 2.67 |
| 398.42 | 4.08 | 4.08 |
| 408.46 | 4.49 | 4.49 |
| 379.85 | 3.88 | 3.88 |
| 409.45 | 4.32 | 4.32 |
| 375.43 | 3.23 | 3.23 |
| 379.85 | 3.88 | 3.88 |
| 392.46 | 5.04 | 5.04 |
| 255.28 | 1.09 | 1.09 |
| 422.49 | 5.05 | 5.05 |
| 376.42 | 3.54 | 3.54 |
| 347.38 | 3.00 | 3.00 |
| 358.40 | 3.33 | 3.33 |
| 375.43 | 3.23 | 3.23 |
| 389.46 | 3.45 | 3.45 |
| 345.41 | 3.23 | 3.23 |
| 392.46 | 5.04 | 5.04 |
| 365.82 | 3.32 | 3.32 |
| 422.49 | 5.05 | 5.05 |