Inhibition of recombinant human CLK1 (130 to end residues) assessed as residual activity at 10 uM using ERMRPRKRQGSVR as substrate incubated for 40 mi...

Basic Information

ID: ALA4815932

Type: Binding

Description: Inhibition of recombinant human CLK1 (130 to end residues) assessed as residual activity at 10 uM using ERMRPRKRQGSVR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control

Format: BAO_0000357

Organism: Homo sapiens

Target:  Dual specificty protein kinase CLK1(ALA4224)

Document:  ALA4813966

Inhibition of recombinant human CLK1 (130 to end residues) assessed as residual activity at 10 uM using ERMRPRKRQGSVR as substrate incubated for 40 mins in presence of [gamma-33ATP] by scintillation counting based radiometry assay relative to control: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
361.412.672.67
436.525.275.27
407.475.095.09
345.413.233.23
331.382.662.66
422.494.884.88
408.464.494.49
361.412.672.67
398.424.084.08
408.464.494.49
379.853.883.88
409.454.324.32
375.433.233.23
379.853.883.88
392.465.045.04
255.281.091.09
422.495.055.05
376.423.543.54
347.383.003.00
358.403.333.33
375.433.233.23
389.463.453.45
345.413.233.23
392.465.045.04
365.823.323.32
422.495.055.05