Basic Information
ID: ALA4821191
Type: Binding
Description: Agonist activity at human GABAB expressed in HEK293T cells co-transfected with human CaV2.2-alpha2delta1 channel assessed as inhibition of CaV2.2-mediated Ba2+ peak-current amplitude at 100 nM at -80 to 10 mV holding potential after 72 hrs by whole cell patch clamp assay relative to control
Organism: Homo sapiens
Cell type: HEK293T
Activity Charts
Bioactivity
Activity Types for Assay ALA4821191
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1766.90 | ||
| 1807.01 | ||
| 1770.93 |