Basic Information
ID: ALA4825222
Type: Binding
Description: Inhibition of N-terminal GST-tagged human recombinant C-KIT V654A mutant (544 to end residues) using GGMEDIYEFMGGKKK as substrate measured after 40 mins in presence of [gamma-33P]ATP by scintillation counting analysis
Format: BAO_0000357
Organism: Homo sapiens
Target: Stem cell growth factor receptor(ALA1936)
Document: ALA4823309
Inhibition of N-terminal GST-tagged human recombinant C-KIT V654A mutant (544 to end residues) using GGMEDIYEFMGGKKK as substrate measured after 40 mins in presence of [gamma-33P]ATP by scintillation counting analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4825222
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 509.62 | 4.06 | 4.06 |
| 411.47 | 3.81 | 3.81 |
| 553.67 | 3.94 | 3.94 |
| 465.57 | 3.21 | 3.21 |
| 412.46 | 3.21 | 3.21 |
| 442.48 | 3.74 | 3.74 |
| 523.60 | 2.91 | 2.91 |
| 480.58 | 3.74 | 3.74 |
| 550.67 | 4.44 | 4.44 |
| 467.53 | 3.97 | 3.97 |
| 367.42 | 3.59 | 3.59 |
| 549.68 | 3.36 | 3.36 |