Basic Information
ID: ALA4828918
Type: Binding
Description: Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane ay 10 uM incubated for 30 mins by microplate beta scintillation counting based radioligand inhibition assay relative to control
Format: BAO_0000249
Organism: Homo sapiens
Cell type: HEK293
Subcellular Fraction: Membrane
Target: Adenosine A2a receptor(ALA251)
Document: ALA4828708
Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HeLa cell membrane ay 10 uM incubated for 30 mins by microplate beta scintillation counting based radioligand inhibition assay relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4828918
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 267.25 | -1.98 | -1.98 |
| 251.25 | -0.95 | -0.95 |
| 399.45 | 0.87 | 0.87 |
| 367.37 | -0.58 | -0.58 |
| 371.40 | -0.19 | -0.19 |
| 371.40 | -0.19 | -0.19 |
| 371.40 | -0.19 | -0.19 |
| 355.40 | 0.83 | 0.83 |
| 367.37 | -0.58 | -0.58 |
| 433.90 | 1.53 | 1.53 |
| 426.48 | 0.63 | 0.63 |
| 417.90 | 2.56 | 2.56 |
| 415.45 | 0.65 | 0.65 |