Inhibition of recombinant GST-Xa-tagged human AAK1 (30 to 330 residues) using 5-FAM-labelled Alla-KEEQSQITSQVTGQIGWR-NH2 peptide as substrate incubate...

Basic Information

ID: ALA4829123

Type: Binding

Description: Inhibition of recombinant GST-Xa-tagged human AAK1 (30 to 330 residues) using 5-FAM-labelled Alla-KEEQSQITSQVTGQIGWR-NH2 peptide as substrate incubated for 3 hrs in presence of ATP by electrophoretic analysis

Format: BAO_0000357

Organism: Homo sapiens

Target: Adaptor-associated kinase(ALA3830)

Document: ALA4828715

Inhibition of recombinant GST-Xa-tagged human AAK1 (30 to 330 residues) using 5-FAM-labelled Alla-KEEQSQITSQVTGQIGWR-NH2 peptide as substrate incubated for 3 hrs in presence of ATP by electrophoretic analysis: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA4829123

IC50

Total(55)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
308.34	3.53	3.53
316.41	2.41	2.41
291.33	2.79	2.79
323.44	3.71	3.71
301.39	3.22	3.22
343.43	3.59	3.59
323.35	2.99	2.99
315.37	2.81	2.81
303.37	1.59	1.59
303.36	2.81	2.81
300.36	3.87	3.87
303.37	1.79	1.79
298.35	2.53	2.53
314.39	2.46	2.46
289.34	2.42	2.42
347.85	3.72	3.72
317.39	3.05	3.05
261.28	1.64	1.64
303.36	2.66	2.66
314.39	2.46	2.46
291.31	1.00	1.00
277.28	0.61	0.61
303.36	2.81	2.81
301.35	2.43	2.43
317.39	2.92	2.92
273.34	2.65	2.65
313.40	3.07	3.07
287.36	2.96	2.96
289.34	2.42	2.42
314.39	2.46	2.46
342.44	3.11	3.11
302.38	2.40	2.40
317.39	3.05	3.05
343.43	3.31	3.31
313.40	3.07	3.07
303.36	2.66	2.66
343.43	3.31	3.31
303.36	2.66	2.66
357.33	3.55	3.55
317.39	2.91	2.91
339.34	3.25	3.25
275.31	2.03	2.03
289.34	2.27	2.27
301.35	2.42	2.42
329.40	3.20	3.20
288.35	3.72	3.72
302.38	2.19	2.19
319.43	3.13	3.13
315.37	2.81	2.81
317.39	2.69	2.69
328.42	2.65	2.65
303.36	2.66	2.66
283.38	3.06	3.06
317.39	3.05	3.05
337.38	2.86	2.86