Basic Information
ID: ALA4829376
Type: Binding
Description: Inhibition of human 20S proteasome LMP2 using Ac-PAL-AMC as fluorogenic substrate measured every minute for 1 hr by fluorescence assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4829376
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 514.62 | 0.73 | 0.73 |
| 578.67 | 0.81 | 0.81 |
| 415.45 | -0.66 | -0.66 |
| 465.59 | 1.33 | 1.33 |
| 465.59 | 1.33 | 1.33 |
| 469.55 | 0.89 | 0.89 |
| 479.62 | 1.72 | 1.72 |
| 465.59 | 1.33 | 1.33 |
| 491.63 | 1.87 | 1.87 |
| 569.74 | 3.72 | 3.72 |
| 485.58 | 1.14 | 1.14 |
| 437.54 | 0.55 | 0.55 |
| 508.62 | 0.06 | 0.06 |
| 451.56 | 0.94 | 0.94 |
| 487.54 | 1.19 | 1.19 |
| 522.64 | 0.45 | 0.45 |
| 595.78 | 4.25 | 4.25 |
| 589.73 | 3.52 | 3.52 |
| 541.69 | 2.94 | 2.94 |
| 555.72 | 3.33 | 3.33 |