Assay Report Card

Basic Information

ID: ALA4829386

Type: Binding

Description: Inhibition of human 20S proteasome LMP2 activity in human NCI/ADR-RES cells overexpressing ABCB1 using Ac-PAL-AMC as fluorogenic substrate incubated for 72 hrs in presence and absence of verapamil by fluorescence assay

Organism: Homo sapiens

Cell type: NCI/ADR-RES

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
589.733.523.52