Basic Information
ID: ALA4831469
Type: Binding
Description: Inhibition of recombinant full length human N-terminal FLAG-tagged PHD1 expressed in baculovirus expression system using HIF1/C35 complex as substrate preincubated for 30 mins followed by substrate addition measured after 10 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4831469
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 345.39 | 3.64 | 3.64 |
| 333.35 | 2.86 | 2.86 |
| 345.36 | 2.64 | 2.64 |
| 340.36 | 1.92 | 1.92 |
| 304.31 | 2.71 | 2.71 |
| 369.41 | 2.27 | 2.27 |