Assay Report Card

Basic Information

ID: ALA4832319

Type: Binding

Description: Inhibition of human KDM4D expressed in Escherichia coli BL21 (DE3) at 1 uM using biotinylated H3-derived peptide and 2-OG as substrate preincubated for 15 mins followed by substrate addition and measured after 1 hr by AlphaLISA assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
417.473.113.11
427.503.253.25
429.523.493.49
435.463.253.25
414.462.602.60
430.483.953.95
381.432.212.21
399.493.483.48
437.503.683.68
478.554.004.00
336.392.222.22
447.493.123.12
489.574.874.87
489.574.874.87
416.482.542.54
418.534.344.34
427.503.553.55
455.493.823.82
413.473.203.20
492.584.304.30
477.564.604.60
461.523.513.51
464.924.604.60
428.562.942.94
414.462.602.60
489.574.874.87
429.523.493.49
369.473.483.48
470.523.603.60
441.533.983.98
435.463.253.25
425.574.774.77
395.462.452.45
417.483.623.62
399.493.483.48
313.361.641.64
429.523.493.49
417.483.623.62
464.924.604.60
489.574.874.87
441.533.653.65
429.523.493.49
437.503.683.68
381.432.212.21
463.534.364.36
479.543.393.39
341.412.242.24
383.452.452.45
397.482.842.84
490.564.274.27
448.474.094.09
488.585.485.48
423.513.383.38
451.913.763.76
489.574.874.87
490.564.274.27
455.493.823.82
489.574.874.87
411.554.604.60
449.453.803.80
438.483.083.08
417.491.761.76
381.432.212.21
461.523.513.51
382.422.632.63
470.523.603.60
447.493.123.12
355.391.821.82
409.533.963.96
467.523.693.69
412.492.782.78