Positive allosteric modulator activity in mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as binding affinity of dyn A1-...

Basic Information

ID: ALA4832456

Type: Binding

Description: Positive allosteric modulator activity in mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as binding affinity of dyn A1-13 to orthosteric binding site at 3 uM coincubated with dyn A1-13 for 90 mins by radioligand competition binding assay

Format: BAO_0000249

Organism: Mus musculus

Cell type: HEK293

Subcellular Fraction: Cell membrane

Target:  Kappa opioid receptor(ALA4329)

Document:  ALA4831505

Positive allosteric modulator activity in mouse kappa opioid receptor stably expressed in HEK293 cell membrane assessed as binding affinity of dyn A1-13 to orthosteric binding site at 3 uM coincubated with dyn A1-13 for 90 mins by radioligand competition binding assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
2937.41