Basic Information
ID: ALA4833083
Type: Binding
Description: Inverse agonist activity at human RORC2 assessed as inhibition of SRC1-derived coactivator peptide by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4833083
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 526.46 | 3.61 | 3.61 |
| 551.47 | 4.14 | 4.14 |
| 566.48 | 3.21 | 3.21 |
| 527.44 | 3.00 | 3.00 |
| 577.50 | 4.12 | 4.12 |
| 524.44 | 3.44 | 3.44 |
| 563.48 | 3.73 | 3.73 |
| 567.51 | 3.78 | 3.78 |
| 524.44 | 3.44 | 3.44 |
| 589.51 | 4.12 | 4.12 |
| 603.54 | 4.23 | 4.23 |
| 549.49 | 4.41 | 4.41 |
| 540.48 | 3.65 | 3.65 |
| 482.40 | 3.19 | 3.19 |
| 538.47 | 3.83 | 3.83 |
| 539.45 | 2.95 | 2.95 |
| 538.47 | 3.49 | 3.49 |
| 568.49 | 3.46 | 3.46 |
| 540.48 | 3.65 | 3.65 |
| 512.43 | 3.22 | 3.22 |
| 550.48 | 3.98 | 3.98 |
| 550.48 | 3.83 | 3.83 |
| 593.55 | 3.55 | 3.55 |
| 543.44 | 3.22 | 3.22 |
| 524.44 | 3.44 | 3.44 |
| 604.53 | 3.62 | 3.62 |
| 510.41 | 3.05 | 3.05 |
| 538.47 | 3.83 | 3.83 |
| 580.50 | 3.60 | 3.60 |
| 594.53 | 3.85 | 3.85 |
| 539.45 | 3.24 | 3.24 |
| 610.56 | 3.68 | 3.68 |
| 554.51 | 3.99 | 3.99 |
| 540.48 | 3.65 | 3.65 |
| 565.49 | 3.48 | 3.48 |
| 554.47 | 3.07 | 3.07 |
| 540.44 | 2.42 | 2.42 |
| 554.47 | 2.81 | 2.81 |
| 540.44 | 3.66 | 3.66 |
| 580.50 | 3.60 | 3.60 |
| 524.44 | 3.44 | 3.44 |
| 581.49 | 2.72 | 2.72 |
| 538.47 | 3.83 | 3.83 |
| 525.43 | 2.56 | 2.56 |
| 564.50 | 4.22 | 4.22 |
| 582.49 | 4.32 | 4.32 |