Assay Report Card

Basic Information

ID: ALA4833715

Type: Functional

Description: Antitumor activity against human KARPAS-422 cells harboring EZH2 Y641N mutant xenografted in NCG mouse assessed as tumor regression at 200 mg/kg, po BID via gavage measured within 10 days

Organism: Homo sapiens

Cell type: KARPAS-422

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
610.804.904.90