Assay Report Card

Basic Information

ID: ALA4833731

Type: Functional

Description: Antitumor activity against human KARPAS-422 cells harboring EZH2 Y641N mutant xenografted in NCG mouse assessed as change in tumor weight at 100 mg/kg, po BID via gavage measured after 28 days (Rvb = 2.14 g)

Organism: Homo sapiens

Cell type: KARPAS-422

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
610.804.904.90