Assay Report Card

Basic Information

ID: ALA4834544

Type: Binding

Description: Inhibition of human PXR expressed in HepG2 cells co-expressing luciferase gene under control of CYP3A4 promoter at 10 uM incubated for 24 hrs by luciferase reporter assay relative to control

Organism: Homo sapiens

Cell type: HepG2

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
410.503.593.59
473.604.484.48
464.394.484.48
431.513.313.31
415.523.723.72
419.934.374.37