Displacement of fluorescent tracer 5-(3-(4-((1S,5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-3-(pyridin-3-ylmethyl)-3,10-diazabicyclo[4.3.1]decan-5-yl...

Basic Information

ID: ALA4835124

Type: Binding

Description: Displacement of fluorescent tracer 5-(3-(4-((1S,5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-3-(pyridin-3-ylmethyl)-3,10-diazabicyclo[4.3.1]decan-5-yl)-1H-1,2,3-triazol-1-yl)propylcarbamoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)benzoate from recombinant full length C-terminal FLAG-tagged FKBP52 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by fluorescence polarisation competition binding assay

Format: BAO_0000219

Organism: Homo sapiens

Target:  FK506 binding protein 4(ALA4050)

Document:  ALA4834405

Displacement of fluorescent tracer 5-(3-(4-((1S,5S,6S)-10-(3,5-dichlorophenylsulfonyl)-2-oxo-3-(pyridin-3-ylmethyl)-3,10-diazabicyclo[4.3.1]decan-5-yl)-1H-1,2,3-triazol-1-yl)propylcarbamoyl)-2-(6-(dimethylamino)-3-(dimethyliminio)-3H-xanthen-9-yl)benzoate from recombinant full length C-terminal FLAG-tagged FKBP52 (unknown origin) expressed in Escherichia coli BL21 (DE3) cells incubated for 30 mins by fluorescence polarisation competition binding assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
715.887.847.84
741.928.408.40
787.998.648.64
787.998.648.64
785.988.428.42
771.958.038.03
701.867.457.45
761.916.186.18
757.927.807.80
701.867.457.45
771.958.038.03
773.968.258.25
771.958.038.03
743.948.628.62
729.918.238.23
741.928.408.40
743.897.417.41
741.928.408.40
771.958.038.03
787.957.437.43
741.928.408.40
727.908.018.01
743.948.628.62
761.916.186.18
727.908.018.01
729.918.238.23
773.968.258.25
727.908.018.01
757.927.807.80
703.877.707.70
785.988.428.42
761.916.186.18
743.897.417.41
715.887.847.84