Assay Report Card

Basic Information

ID: ALA4836049

Type: Binding

Description: Inhibition of human ERG expressed in CHO cells at 30 uM with holding potential at -80 to -60 mV for 500s followed by raise in potential at +30 mV for 2 sec and subsequent repolarization to -60 mV for 2 sec by whole-cell patch clamp method relative to control

Organism: Homo sapiens

Cell type: CHO

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
472.176.126.12
388.504.924.92
350.454.344.34
343.434.314.31
380.305.175.17