ID: ALA4836378
Type: Binding
Description: Displacement of Alexafluor 647-conjugated PFI-1 from N-terminal-His6-tagged human BRD4 BD1 domain (44 to 170 residues) incubated for 30 mins by fluorescence polarization assay
Format: BAO_0000357
Organism: Homo sapiens
Target: Bromodomain-containing protein 4(ALA1163125)
Document: ALA4834448
Displacement of Alexafluor 647-conjugated PFI-1 from N-terminal-His6-tagged human BRD4 BD1 domain (44 to 170 residues) incubated for 30 mins by fluorescence polarization assay: 1
Bioactivity
Activity Types for Assay ALA4836378
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
220.28 | 0.09 | 0.09 |
274.37 | 1.26 | 1.26 |
260.35 | 1.08 | 1.08 |
288.40 | 1.64 | 1.64 |