Basic Information
ID: ALA4836549
Type: Binding
Description: Binding affinity to 6His-Thr-BRD4 (1 to 477 residues) BD2 domain Y390A mutant (unknown origin) incubated for 30 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4836549
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 491.56 | 5.06 | 5.06 |
| 325.37 | 1.15 | 1.15 |
| 414.48 | 3.96 | 3.96 |
| 410.45 | 2.28 | 2.28 |
| 339.40 | 1.71 | 1.71 |
| 364.41 | 1.63 | 1.63 |
| 356.43 | 1.76 | 1.76 |
| 404.89 | 3.48 | 3.48 |
| 438.45 | 2.90 | 2.90 |
| 354.41 | 2.17 | 2.17 |
| 384.48 | 2.19 | 2.19 |
| 330.39 | 0.96 | 0.96 |
| 314.39 | 2.93 | 2.93 |
| 400.48 | 2.83 | 2.83 |
| 404.89 | 3.48 | 3.48 |
| 312.37 | 2.68 | 2.68 |
| 370.45 | 1.89 | 1.89 |
| 404.90 | 2.54 | 2.54 |
| 368.43 | 2.29 | 2.29 |
| 438.45 | 2.90 | 2.90 |
| 368.44 | 1.35 | 1.35 |
| 384.48 | 3.13 | 3.13 |
| 384.48 | 3.13 | 3.13 |
| 314.39 | 1.99 | 1.99 |
| 316.36 | 1.51 | 1.51 |
| 339.40 | 1.71 | 1.71 |
| 404.90 | 2.54 | 2.54 |
| 382.46 | 2.01 | 2.01 |
| 404.90 | 2.54 | 2.54 |
| 316.36 | 0.57 | 0.57 |
| 384.48 | 2.54 | 2.54 |
| 404.89 | 3.48 | 3.48 |
| 370.45 | 2.82 | 2.82 |
| 400.48 | 1.51 | 1.51 |
| 384.48 | 3.48 | 3.48 |
| 382.46 | 1.74 | 1.74 |
| 330.38 | 1.90 | 1.90 |
| 382.46 | 1.74 | 1.74 |
| 286.34 | 1.21 | 1.21 |
| 312.37 | 1.74 | 1.74 |
| 402.88 | 2.00 | 2.00 |
| 180.21 | 0.97 | 0.97 |
| 402.88 | 2.00 | 2.00 |
| 312.37 | 2.68 | 2.68 |
| 300.36 | 1.60 | 1.60 |
| 300.36 | 2.54 | 2.54 |
| 388.44 | 2.96 | 2.96 |
| 384.48 | 2.28 | 2.28 |
| 298.35 | 1.18 | 1.18 |