Basic Information
ID: ALA4836630
Type: Binding
Description: Inhibition of 6His-Thr-BRD4 (1 to 477 residues) BD2 domain Y390A mutant (unknown origin) incubated for 30 mins by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA4836630
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 342.37 | 2.27 | 2.27 |
| 471.53 | 2.12 | 2.12 |
| 325.37 | 1.15 | 1.15 |
| 410.45 | 2.28 | 2.28 |
| 368.41 | 2.80 | 2.80 |
| 328.34 | 2.01 | 2.01 |
| 364.45 | 2.88 | 2.88 |
| 396.42 | 2.08 | 2.08 |
| 324.38 | 2.10 | 2.10 |
| 366.42 | 2.47 | 2.47 |
| 392.46 | 2.12 | 2.12 |
| 380.44 | 1.86 | 1.86 |
| 336.39 | 2.46 | 2.46 |
| 406.48 | 2.24 | 2.24 |
| 408.50 | 2.78 | 2.78 |
| 386.45 | 1.32 | 1.32 |
| 392.46 | 2.07 | 2.07 |
| 376.42 | 2.56 | 2.56 |
| 379.42 | 1.34 | 1.34 |
| 310.35 | 1.93 | 1.93 |
| 439.51 | 1.78 | 1.78 |
| 404.47 | 2.28 | 2.28 |
| 379.42 | 1.34 | 1.34 |
| 392.46 | 2.25 | 2.25 |
| 354.38 | 2.60 | 2.60 |
| 296.33 | 1.67 | 1.67 |
| 443.51 | 2.76 | 2.76 |
| 382.44 | 3.05 | 3.05 |
| 378.43 | 1.95 | 1.95 |
| 433.51 | 2.17 | 2.17 |
| 379.42 | 1.34 | 1.34 |
| 406.48 | 2.24 | 2.24 |
| 375.43 | 2.94 | 2.94 |
| 354.38 | 2.60 | 2.60 |
| 408.45 | 1.95 | 1.95 |
| 350.42 | 2.64 | 2.64 |
| 417.47 | 2.43 | 2.43 |
| 408.45 | 1.09 | 1.09 |
| 350.42 | 2.71 | 2.71 |
| 406.48 | 2.51 | 2.51 |