ID: ALA4836631
Type: Binding
Description: Inhibition of 6His-Thr-BRD4 (1 to 477 residues) BD1 domain (unknown origin) incubated for 30 mins by TR-FRET assay
Organism: Homo sapiens
Bioactivity
Activity Types for Assay ALA4836631
IC50
Parent Molecular Weight | ALogP | Polar Surface Area |
---|---|---|
342.37 | 2.27 | 2.27 |
471.53 | 2.12 | 2.12 |
325.37 | 1.15 | 1.15 |
410.45 | 2.28 | 2.28 |
368.41 | 2.80 | 2.80 |
328.34 | 2.01 | 2.01 |
364.45 | 2.88 | 2.88 |
396.42 | 2.08 | 2.08 |
324.38 | 2.10 | 2.10 |
366.42 | 2.47 | 2.47 |
392.46 | 2.12 | 2.12 |
380.44 | 1.86 | 1.86 |
336.39 | 2.46 | 2.46 |
406.48 | 2.24 | 2.24 |
408.50 | 2.78 | 2.78 |
386.45 | 1.32 | 1.32 |
392.46 | 2.07 | 2.07 |
376.42 | 2.56 | 2.56 |
379.42 | 1.34 | 1.34 |
310.35 | 1.93 | 1.93 |
439.51 | 1.78 | 1.78 |
404.47 | 2.28 | 2.28 |
379.42 | 1.34 | 1.34 |
392.46 | 2.25 | 2.25 |
354.38 | 2.60 | 2.60 |
296.33 | 1.67 | 1.67 |
443.51 | 2.76 | 2.76 |
382.44 | 3.05 | 3.05 |
378.43 | 1.95 | 1.95 |
433.51 | 2.17 | 2.17 |
379.42 | 1.34 | 1.34 |
406.48 | 2.24 | 2.24 |
375.43 | 2.94 | 2.94 |
354.38 | 2.60 | 2.60 |
408.45 | 1.95 | 1.95 |
350.42 | 2.64 | 2.64 |
417.47 | 2.43 | 2.43 |
408.45 | 1.09 | 1.09 |
350.42 | 2.71 | 2.71 |
406.48 | 2.51 | 2.51 |