Inhibition of wild type HIV1 protease using Arg-Glu (EDANS)-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincubated for 20 to 30 min...

Basic Information

ID: ALA4837920

Type: Binding

Description: Inhibition of wild type HIV1 protease using Arg-Glu (EDANS)-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincubated for 20 to 30 mins followed by substrate addition and measured for 10 mins by FRET assay

Format: BAO_0000357

Organism: Human immunodeficiency virus 1

Target:  Human immunodeficiency virus type 1 protease(ALA243)

Document:  ALA4837199

Inhibition of wild type HIV1 protease using Arg-Glu (EDANS)-Ser-Gln-Asn-Tyr-Pro-Ile-Val-Gln-Lys(DABCYL)-Arg as substrate preincubated for 20 to 30 mins followed by substrate addition and measured for 10 mins by FRET assay: 1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
547.672.382.38
555.663.443.44
502.682.152.15
502.682.002.00
555.663.443.44
555.663.583.58
585.694.054.05
555.663.443.44
517.692.572.57
502.682.002.00
569.693.783.78
531.722.772.77
516.712.352.35
532.712.612.61
532.712.612.61
502.682.002.00
547.723.043.04
547.723.043.04
517.692.432.43
585.694.054.05
517.692.432.43
517.692.432.43