Basic Information
ID: ALA4843621
Type: Binding
Description: Inhibition of recombinant CETP (unknown origin) assessed as maximal inhibition of transfer of [3H]cholesteryl oleate or [3H]triolein using exogenous LDL and HDL in 2% human serum at 10 uM measured after 2 hrs by liquid scintillation analysis relative to control
Format: BAO_0000357
Organism: Homo sapiens
Target: Cholesteryl ester transfer protein(ALA3572)
Document: ALA4842348
Inhibition of recombinant CETP (unknown origin) assessed as maximal inhibition of transfer of [3H]cholesteryl oleate or [3H]triolein using exogenous LDL and HDL in 2% human serum at 10 uM measured after 2 hrs by liquid scintillation analysis relative to control: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4843621
Imax
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 619.52 | 9.62 | 9.62 |
| 637.51 | 9.76 | 9.76 |
| 697.55 | 9.87 | 9.87 |
| 653.54 | 10.17 | 10.17 |
| 697.55 | 9.87 | 9.87 |
| 667.57 | 10.48 | 10.48 |
| 711.58 | 10.17 | 10.17 |
| 671.53 | 10.31 | 10.31 |
| 716.00 | 10.82 | 10.82 |
| 641.93 | 10.41 | 10.41 |