Assay Report Card

Basic Information

ID: ALA4844394

Type: Binding

Description: Protac activity at VHL/AR T878A mutant in human LNCaP cells assessed as reduction in AR protein level at 100 nM measured after 6 hrs by western blot analysis

Organism: Homo sapiens

Cell type: LNCaP

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
792.344.484.48
806.365.025.02
820.395.265.26
820.395.265.26
806.365.025.02