Basic Information
ID: ALA4844510
Type: Functional
Description: Antagonist activity at human 5HT6R expressed in 1321N1 cells assessed as inhibition of IBMX-induced cAMP production measured after 30 mins by TR-FRET assay
Format: BAO_0000219
Organism: Homo sapiens
Cell type: 1321N1
Target: Serotonin 6 (5-HT6) receptor(ALA3371)
Document: ALA4842370
Antagonist activity at human 5HT6R expressed in 1321N1 cells assessed as inhibition of IBMX-induced cAMP production measured after 30 mins by TR-FRET assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA4844510
Kb
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 487.36 | 2.85 | 2.85 |
| 550.68 | 4.09 | 4.09 |
| 517.57 | 4.66 | 4.66 |
| 568.74 | 6.17 | 6.17 |
| 449.58 | 3.64 | 3.64 |
| 484.02 | 4.29 | 4.29 |