Assay Report Card

Basic Information

ID: ALA5030475

Type: Binding

Description: Antagonist activity at human RXR-alpha expressed in African green monkey COS-1 cells assessed as reduction in NEt-TMN-induced receptor transactivation by measuring shift in concentration-response curve at 1 uM by luciferase reporter gene assay

Organism: Homo sapiens

Cell type: COS-1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
439.606.256.25
504.556.516.51
449.606.436.43
435.576.046.04
502.587.667.66
516.608.058.05