Assay Report Card

Basic Information

ID: ALA5032407

Type: Binding

Description: Inhibition of human N-terminal His6-tagged KDM3B (L882 to S1761 residues) expressed in insect cells using H3K9(Me2) as substrate preincubated for 15 mins followed by substrate addition and measured after 5 mins by Alphascreen assay

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
290.342.192.19
242.301.751.75
270.270.640.64
268.342.142.14
262.291.761.76
172.160.130.13
290.301.441.44
228.271.361.36
242.210.160.16
276.321.801.80
186.190.190.19
304.372.582.58
298.413.313.31