Basic Information
ID: ALA5033965
Type: Functional
Description: Agonist activity at human RXFP1 expressed in human CHO-K1 cells assessed as inhibition of H2 relaxin-induced cAMP accumulation at 10 uM incubated for 30 mins by TR-FRET assay relative to H2 relaxin
Format: BAO_0000219
Organism: Homo sapiens
Cell type: CHO-K1
Target: Relaxin receptor 1(ALA1293316)
Document: ALA5032539
Agonist activity at human RXFP1 expressed in human CHO-K1 cells assessed as inhibition of H2 relaxin-induced cAMP accumulation at 10 uM incubated for 30 mins by TR-FRET assay relative to H2 relaxin: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5033965
Activity
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 383.88 | 3.78 | 3.78 |
| 383.88 | 3.83 | 3.83 |
| 407.47 | 2.96 | 2.96 |
| 350.43 | 2.57 | 2.57 |
| 475.33 | 3.78 | 3.78 |
| 379.46 | 3.18 | 3.18 |
| 350.43 | 2.57 | 2.57 |
| 355.47 | 3.24 | 3.24 |
| 378.87 | 3.69 | 3.69 |
| 394.44 | 3.08 | 3.08 |
| 367.43 | 3.31 | 3.31 |
| 397.91 | 4.08 | 4.08 |
| 388.48 | 3.30 | 3.30 |
| 392.51 | 3.24 | 3.24 |
| 381.46 | 3.57 | 3.57 |
| 364.45 | 2.82 | 2.82 |
| 428.33 | 3.94 | 3.94 |
| 350.43 | 2.57 | 2.57 |
| 402.46 | 2.83 | 2.83 |
| 355.47 | 3.24 | 3.24 |
| 359.44 | 2.69 | 2.69 |
| 374.45 | 3.05 | 3.05 |