Assay Report Card

Basic Information

ID: ALA5039019

Type: Binding

Description: Binding affinity to EZH2 in human WSUDLCL2 cells assessed as thermal stability by measuring shift in temperature at 60 uM pretreated with proteasome inhibitor MG132 for 1 hr followed by compound addition incubated for 2 hrs by cellular thermal shift based Western blot analysis

Organism: Homo sapiens

Cell type: WSUDLCL2

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
942.176.456.45