Assay Report Card

Basic Information

ID: ALA5039145

Type: Binding

Description: Selectivity index, ratio of IC50 for inhibition of recombinant full length human N-terminal FLAG-tagged EZH1 in PRC2 complex expressed in baculovirus system to IC50 for inhibition of N-terminal His-tagged EZH2 in human PCR2 complex (2 to end residues) expressed in Sf9 cells

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
942.176.456.45