Assay Report Card

Basic Information

ID: ALA5039702

Type: Binding

Description: Inhibition of human ABL Q252H mutant using EAIYAAPFAKKK as substrate assessed as residual activity at 10 nM incubated for 30 mins followed by 33P-ATP addition and measured after 2 hrs by liquid scintillation counter method relative to control

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
532.574.464.46
526.594.474.47