Basic Information
ID: ALA5042806
Type: Binding
Description: Inhibition of DYRK1A (unknown origin) using Ulight-MBP as substrate and ATP as co-substrate incubated for 40 mins and measured after 1 hr by TR-FRET assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5042806
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 212.25 | 3.03 | 3.03 |
| 216.24 | 1.32 | 1.32 |
| 280.34 | 2.30 | 2.30 |
| 374.45 | 3.43 | 3.43 |
| 296.33 | 2.23 | 2.23 |
| 322.29 | 2.53 | 2.53 |
| 374.45 | 3.43 | 3.43 |
| 240.27 | 2.36 | 2.36 |
| 350.47 | 3.94 | 3.94 |
| 348.38 | 3.15 | 3.15 |
| 253.30 | 3.28 | 3.28 |
| 334.38 | 2.80 | 2.80 |
| 200.24 | 2.34 | 2.34 |
| 361.41 | 2.44 | 2.44 |
| 304.30 | 2.23 | 2.23 |
| 203.67 | 3.71 | 3.71 |
| 234.69 | 2.99 | 2.99 |
| 375.44 | 2.83 | 2.83 |
| 195.22 | 3.49 | 3.49 |
| 350.35 | 3.31 | 3.31 |
| 240.27 | 1.19 | 1.19 |
| 226.24 | 0.96 | 0.96 |
| 226.24 | 2.05 | 2.05 |
| 296.38 | 2.77 | 2.77 |
| 239.28 | 3.12 | 3.12 |
| 210.24 | 3.08 | 3.08 |
| 239.28 | 1.80 | 1.80 |
| 224.26 | 3.39 | 3.39 |
| 335.43 | 4.79 | 4.79 |
| 454.33 | 3.59 | 3.59 |
| 308.39 | 3.08 | 3.08 |
| 228.25 | 1.24 | 1.24 |
| 279.34 | 2.90 | 2.90 |
| 226.24 | 0.96 | 0.96 |
| 226.24 | 2.05 | 2.05 |
| 297.36 | 3.53 | 3.53 |
| 360.42 | 3.05 | 3.05 |
| 254.30 | 1.50 | 1.50 |
| 241.32 | 3.13 | 3.13 |
| 440.31 | 3.20 | 3.20 |
| 253.26 | 2.02 | 2.02 |
| 312.38 | 2.00 | 2.00 |
| 236.28 | 2.46 | 2.46 |
| 226.24 | 2.05 | 2.05 |
| 259.70 | 3.31 | 3.31 |
| 338.46 | 3.80 | 3.80 |
| 225.25 | 1.56 | 1.56 |
| 225.25 | 2.66 | 2.66 |
| 226.24 | 2.05 | 2.05 |
| 310.41 | 3.02 | 3.02 |
| 375.44 | 2.83 | 2.83 |
| 242.31 | 2.52 | 2.52 |
| 395.85 | 3.09 | 3.09 |
| 245.28 | 0.98 | 0.98 |
| 227.27 | 1.85 | 1.85 |
| 296.38 | 2.72 | 2.72 |
| 199.25 | 3.07 | 3.07 |
| 239.28 | 2.97 | 2.97 |