Assay Report Card

Basic Information

ID: ALA5042938

Type: Binding

Description: Protac activity at VHL/EZH2 in human 22Rv1 cells assessed as reduction in EZH2 level at 2 uM preincubated with VH032 for 2 hrs followed by compound addition and measured after 24 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: 22Rv1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1048.32