Assay Report Card

Basic Information

ID: ALA5042943

Type: Binding

Description: Protac activity at VHL/EZH2 in human 22Rv1 cells assessed as reduction in H3K27me3 level at 1 uM incubated for 48 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: 22Rv1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1163.45
1119.40
1075.34
1048.32
1018.29