Basic Information
ID: ALA5045604
Type: Binding
Description: Inhibition of fluorescent antagonist binding to mouse P2Y14R expressed in HEK293 cells preincubated for 30 mins followed by addition of 6-amino-9-(2-carboxy-4-((6-(4-(4-(4-(4-(3-carboxy-6-(4-(trifluoromethyl)phenyl)naphthalen-1-yl)phenyl)piperidin-1-yl)butyl)-1H-1,2,3-triazol-1-yl)hexyl)carbamoyl)phenyl)-3-iminio-5-sulfo-3H-xanthene-4-sulfonate incubated for 30 mins by BD FACSCalibur flow cytometry analysis
Organism: Mus musculus
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5045604
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 487.52 | 7.36 | 7.36 |
| 501.50 | 6.88 | 6.88 |
| 519.52 | 6.80 | 6.80 |
| 517.55 | 6.71 | 6.71 |
| 505.54 | 6.70 | 6.70 |
| 501.50 | 6.88 | 6.88 |
| 487.52 | 7.36 | 7.36 |
| 487.52 | 7.36 | 7.36 |
| 564.62 | 7.82 | 7.82 |
| 529.56 | 7.62 | 7.62 |