Displacement of Alexafluor 647-JQ1 from GST-BRD4 BD1 BD2 (44 to 460 residues) (unknown origin) incubated for 60 mins by fluorescence polarization assa...

Basic Information

ID: ALA5045654

Type: Binding

Description: Displacement of Alexafluor 647-JQ1 from GST-BRD4 BD1 BD2 (44 to 460 residues) (unknown origin) incubated for 60 mins by fluorescence polarization assay

Format: BAO_0000357

Organism: Homo sapiens

Target: Bromodomain-containing protein 4(ALA1163125)

Document: ALA5042544

Displacement of Alexafluor 647-JQ1 from GST-BRD4 BD1 BD2 (44 to 460 residues) (unknown origin) incubated for 60 mins by fluorescence polarization assay: 1

Associated Items: Associated Bioactivities Associated Compounds

Activity Charts

Bioactivity

Activity Types for Assay ALA5045654

IC50

Total(20)

Compound Summary

Parent Molecular Weight	ALogP	Polar Surface Area
368.39	1.65	1.65
426.48	2.65	2.65
362.39	0.86	0.86
460.54	1.18	1.18
562.69	3.32	3.32
412.45	2.26	2.26
323.35	0.92	0.92
362.39	1.10	1.10
338.37	0.21	0.21
363.38	0.25	0.25
474.57	1.57	1.57
510.47	3.54	3.54
376.42	2.12	2.12
516.65	2.59	2.59
566.66	3.23	3.23
368.39	1.65	1.65
376.42	1.45	1.45
459.55	1.78	1.78
454.53	3.28	3.28
566.66	3.23	3.23