Assay Report Card

Basic Information

ID: ALA5046678

Type: Binding

Description: Protac activity at CDK2/VHL E3 ligase in human HEI-OC1 cells assessed as induction of CDK2 protein degradation at 100 nM measured after 24 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: HEI-OC1

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
371.473.383.38
382.252.452.45
960.084.054.05
981.225.235.23