Basic Information
ID: ALA5049597
Type: Binding
Description: Inhibition of GST-Xa tagged human AAK1 (30 to 330 residues) expresssed in bacteria using (5-FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 peptide as substrate incubated for 3 hrs in presence of ATP by electrophoretic analysis
Format: BAO_0000357
Organism: Homo sapiens
Target: Adaptor-associated kinase(ALA3830)
Document: ALA5046296
Inhibition of GST-Xa tagged human AAK1 (30 to 330 residues) expresssed in bacteria using (5-FAM)-Aha-KEEQSQITSQVTGQIGWR-NH2 peptide as substrate incubated for 3 hrs in presence of ATP by electrophoretic analysis: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5049597
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 289.34 | 2.27 | 2.27 |
| 366.43 | 5.22 | 5.22 |
| 349.43 | 4.53 | 4.53 |
| 352.40 | 4.91 | 4.91 |
| 333.86 | 4.25 | 4.25 |
| 360.41 | 4.10 | 4.10 |
| 324.43 | 3.47 | 3.47 |
| 270.38 | 3.50 | 3.50 |
| 363.38 | 4.39 | 4.39 |
| 369.84 | 4.88 | 4.88 |
| 270.38 | 3.50 | 3.50 |
| 349.42 | 4.53 | 4.53 |
| 402.41 | 5.85 | 5.85 |
| 369.84 | 4.88 | 4.88 |
| 359.42 | 4.70 | 4.70 |
| 349.42 | 4.53 | 4.53 |
| 309.41 | 3.68 | 3.68 |
| 323.44 | 4.07 | 4.07 |
| 333.86 | 4.25 | 4.25 |
| 369.84 | 4.88 | 4.88 |
| 370.39 | 5.05 | 5.05 |
| 384.42 | 5.77 | 5.77 |
| 313.44 | 3.90 | 3.90 |
| 333.86 | 4.25 | 4.25 |
| 338.50 | 5.08 | 5.08 |
| 325.41 | 3.38 | 3.38 |
| 385.41 | 5.16 | 5.16 |
| 348.44 | 5.14 | 5.14 |
| 374.48 | 5.71 | 5.71 |