Basic Information
ID: ALA5054769
Type: Binding
Description: Bump and hole PROTAC activity at BromoTag-Brd2/VHL-bound E3 ligase in HEK293 cells assessed as Brd2 degradation at 0.001 to 10 uM measured after 6 hrs by Western blot analysis
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5054769
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1000.69 | ||
| 1015.70 | ||
| 1030.71 | ||
| 1017.67 | ||
| 1031.70 | ||
| 1014.72 | ||
| 1015.70 | ||
| 1031.70 | ||
| 1016.69 | ||
| 1030.71 | ||
| 1001.67 |