Assay Report Card

Basic Information

ID: ALA5054770

Type: Binding

Description: Bump and hole PROTAC activity at BromoTag-Brd2 BD2 L387A mutant/VHL-bound E3 ligase in HEK293 cells assessed as Brd2 degradation measured after 6 hrs by Western blot analysis

Organism: Homo sapiens

Cell type: HEK293

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
1000.69
1015.70
1030.71
1017.67
1031.70
1014.72
1015.70
1031.70
1016.69
1030.71
1001.67