Basic Information
ID: ALA5054780
Type: Binding
Description: Reversibility of Bump and hole PROTAC activity at BromoTag-Brd2 BD2 L387A mutant/VHL-bound E3 ligase in HEK293 cells assessed as Brd2 degradation at 200 nM treated for 3 hrs measured after 24 hrs of compound washout by Western blot analysis
Organism: Homo sapiens
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5054780
Inhibition
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1031.70 |