Assay Report Card

Basic Information

ID: ALA5097988

Type: Binding

Description: Selectivity index, ratio of IC50 for Inhibition of full length N-terminal GST-tagged human recombinant HDAC7 (501 to 952 residues) expressed in Baculovirus system using Ac-Leu-Gly-Lys (Ac)-AMC as substrate to IC50 for inhibition of recombinant HDAC3 (unknown origin) using Ac-Leu-Gly-Lys (Ac)-AMC as substrate pretreated

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
588.695.795.79
602.716.186.18
574.665.405.40
546.614.624.62
515.595.305.30
589.716.626.62
518.604.704.70
532.625.095.09
472.523.733.73
520.564.764.76
616.746.576.57
541.635.425.42
546.605.165.16