Assay Report Card

Basic Information

ID: ALA5097990

Type: Binding

Description: Selectivity index, ratio of IC50 for Inhibition of full length N-terminal GST-tagged human recombinant HDAC7 (501 to 952 residues) expressed in Baculovirus system using Ac-Leu-Gly-Lys (Ac)-AMC as substrate to IC50 for inhibition of full length N-terminal GST-tagged human recombinant HDAC6 (1 to 1215 residues) expressed in Baculovirus infected Sf9 cells using Ac-Leu-Gly-Lys (Ac)-AMC as substrate

Organism: Homo sapiens

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
483.503.073.07
513.574.074.07
440.483.593.59
527.604.464.46
499.553.683.68
485.523.293.29