Assay Report Card

Basic Information

ID: ALA5098707

Type: Binding

Description: Inhibition of CDK9 in human MCF7 cells assessed as reduction in RNA polymerase II phosphorylation at ser2 residue preincubated for 6 hrs followed by compound washout and measured at 2 to 4 hrs by fluorescence based assay

Organism: Homo sapiens

Cell type: MCF7

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
461.614.164.16
447.583.773.77