Basic Information
ID: ALA5099275
Type: Binding
Description: Inhibition of CA200645 binding to NanoLuc-fused rat adenosine A1 receptor expressed in HEK293 cells assessed as kinetic dissociation constant by NanoBRET competition binding assay
Organism: Rattus norvegicus
Cell type: HEK293
Activity Charts
Bioactivity
Activity Types for Assay ALA5099275
Kd
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 267.25 | -1.98 | -1.98 |
| 308.30 | -1.84 | -1.84 |
| 441.49 | 0.99 | 0.99 |
| 512.57 | 1.14 | 1.14 |
| 468.51 | 0.99 | 0.99 |
| 483.57 | 2.15 | 2.15 |
| 561.44 | 1.89 | 1.89 |
| 506.36 | 1.61 | 1.61 |
| 502.96 | 1.65 | 1.65 |
| 520.38 | 1.75 | 1.75 |
| 520.38 | 1.75 | 1.75 |
| 516.99 | 1.78 | 1.78 |
| 427.46 | 0.85 | 0.85 |
| 461.91 | 1.50 | 1.50 |
| 498.54 | 1.00 | 1.00 |
| 471.51 | 1.00 | 1.00 |
| 524.62 | 2.29 | 2.29 |
| 502.96 | 1.65 | 1.65 |
| 502.96 | 1.65 | 1.65 |
| 461.91 | 1.50 | 1.50 |
| 475.93 | 1.64 | 1.64 |
| 457.49 | 0.86 | 0.86 |
| 547.41 | 1.76 | 1.76 |
| 461.91 | 1.50 | 1.50 |
| 561.44 | 1.89 | 1.89 |
| 516.99 | 1.78 | 1.78 |
| 475.93 | 1.64 | 1.64 |