Basic Information
ID: ALA5100331
Type: Binding
Description: Inhibition of wild type partial length human PDGFRbeta (V582 to Y1009 residues) expressed in bacterial expression system using Ulight-p70S6K peptide substrate incubated for 90 mins in presence of ATP by HTRF assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5100331
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 454.44 | 2.60 | 2.60 |
| 486.45 | 3.40 | 3.40 |
| 460.54 | 3.68 | 3.68 |
| 418.46 | 2.32 | 2.32 |
| 362.39 | 2.17 | 2.17 |
| 380.38 | 2.30 | 2.30 |
| 450.47 | 2.77 | 2.77 |
| 419.45 | 1.72 | 1.72 |