Assay Report Card

Basic Information

ID: ALA5106121

Type: Binding

Description: Displacement of [3H]ZM241385 from human adenosine A2A receptor expressed in HEK293 cell membrane at 1 uM preincubated for 4 hrs followed by [3H]ZM241385 addition and measured after 0.5 hrs by radioligand displacement assay

Organism: Homo sapiens

Cell type: HEK293

Subcellular Fraction: Cell membrane

Activity Charts

Compound Summary

Parent Molecular WeightALogPPolar Surface Area
394.432.032.03
410.431.971.97
369.453.113.11
410.431.971.97
368.351.081.08
352.351.151.15
369.453.113.11
394.432.032.03
368.351.081.08
352.351.151.15
327.372.222.22
327.372.222.22