Basic Information
ID: ALA5108379
Type: Binding
Description: Displacement of (2S,4R)-N-(4-bromobenzyl)-4-hydroxy-1-(3,3,3-trifluoropropanoyl)pyrrolidine-2-carboxamide from BRD4 bromodomain 2/VBC E3 ligase (unknown origin) ternary complex assessed as inhibition constant by 19F NMR assay
Organism: Homo sapiens
Activity Charts
Bioactivity
Activity Types for Assay ALA5108379
Ki
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 1080.75 | ||
| 1002.66 | ||
| 992.64 | 7.31 | 7.31 |
| 1036.69 | ||
| 1020.65 |