Basic Information
ID: ALA5112650
Type: Binding
Description: Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) incubated for 30 mins by Alphascreen assay
Format: BAO_0000019
Organism: Homo sapiens
Target: Protein polybromo-1(ALA1795184)
Document: ALA5108070
Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) incubated for 30 mins by Alphascreen assay: 1
Activity Charts
Bioactivity
Activity Types for Assay ALA5112650
IC50
Compound Summary
| Parent Molecular Weight | ALogP | Polar Surface Area |
|---|---|---|
| 239.23 | 2.38 | 2.38 |
| 291.69 | 3.48 | 3.48 |
| 238.29 | 2.85 | 2.85 |
| 302.80 | 4.27 | 4.27 |
| 273.67 | 3.03 | 3.03 |
| 258.71 | 3.19 | 3.19 |
| 272.74 | 3.50 | 3.50 |
| 288.73 | 3.20 | 3.20 |
| 276.70 | 3.33 | 3.33 |
| 291.69 | 3.48 | 3.48 |
| 311.14 | 3.98 | 3.98 |
| 252.32 | 3.16 | 3.16 |
| 256.28 | 2.99 | 2.99 |
| 317.19 | 3.61 | 3.61 |
| 300.79 | 4.12 | 4.12 |
| 317.19 | 3.61 | 3.61 |
| 273.68 | 3.03 | 3.03 |
| 286.76 | 3.81 | 3.81 |
| 286.76 | 3.81 | 3.81 |
| 286.76 | 3.81 | 3.81 |
| 272.74 | 3.50 | 3.50 |
| 272.74 | 3.50 | 3.50 |
| 286.76 | 3.81 | 3.81 |
| 270.72 | 3.55 | 3.55 |
| 293.15 | 3.85 | 3.85 |
| 268.32 | 2.86 | 2.86 |
| 271.70 | 3.82 | 3.82 |
| 326.70 | 4.21 | 4.21 |
| 311.14 | 3.99 | 3.99 |
| 276.70 | 3.33 | 3.33 |
| 268.36 | 3.62 | 3.62 |
| 286.76 | 3.81 | 3.81 |